Our Science

Our Science : Patents

  1. Bair, K. W.; Herbertz, T.; Kauffman, G. S.; Kayser-Bricker, K. J.; Luke, G. P.; Martin, M. W.; Millan, D. S.; Schiller, S. E. R.; Talbot, A. C. “Tetrahydroquinoline compositions as BET bromodomain inhibitors and their preparation” WO 2015074064, 2015.

  2. Bair, K. W.; Herbertz, T.; Kauffman, G. S.; Kayser-Bricker, K. J.; Luke, G. P.; Martin, M. W.; Millan, D. S.; Schiller, S. E. R.; Talbot, A. C.; Tebb, M. J.. “Benzopiperazine compositions as BET bromodomain inhibitors and their preparation” WO 2015074081, 2015.

  3. Bair, K. W.; Millan, D. S.; Martin, M. W.; Tebbe, M. J.; Lu, W.; Li, H.; Loch, J. “Preparation of FASN inhibitors useful for treatment of cancer and other diseases” WO 2014164767, 2014.

  4. Bair, K. W.; Lancia, D. R.; Li, H.; Loch, J.; Lu, W.; Martin, M. W.; Millan, D. S.; Schiller, S. E. R.; Tebbe, M. J. “Preparation of biarylcarbonylpiperazinylcarbonylcycloalkanol derivatives as FASN inhibitors for treatment of cancer and other diseases” WO 2014164749, 2014.

  5. Bair, K. W.; Baumeister, T. R.; Dragovich, P.; Zak, M.; Zhao, G.; Zheng, X. “Cyclopropanecarboxamide derivatives as NAMPT inhibitors and their preparation” WO 2014074715, 2014.

  6. Bair, K. W.; Baumeister, T. R.; Gosselin, F.; Zak, M.; Zheng, X. “Amido-benzyl sulfoxide derivatives” WO 2013130935, 2013.

  7. Bair, K. W.; Baumeister, T. R.; Buckmelter, A. J.; Clodfelter, K. H.; Gunzner-Toste, J.; Han, B.; Lin, J.; Reynolds, D. J.; Smith, C. C.; Wang, Z.; Zak, M.; Zheng, X.; Zhao, G. “Alkyl-and di-substituted amido-benzyl sulfonamide derivatives” WO 2013130943, 2013.

  8. Yuen, P-W.; Bair, K. W.; Baumeister, T. R.; Dragovich, P.; Liu, X.; Patel, S.; Zak, M.; Zhao, G.; Zhang, Y.; Zheng, X. “Amido spirocyclic amide and sulfonamide derivatives” WO 2013127269, 2013.

  9. Bair, K. W.; Baumeister, T. R.; Buckmelter, A. J.; Clodfelter, K. H.; Dragovich, P.; Gosselin, F.; Gunzner-Toste, J.; Han, B.; Lin, J.; Liu, X.; Reynolds, D. J.; Smith, C. C.; Wang, Z.; Zak, M.; Zhang, Y.; Zhao, G.; Zheng, X.; Yuen, P-W. “Amido-benzyl sulfone and sulfoxide derivatives” WO 2013127266, 2013.

  10. Bair, K. W.; Baumeister, T. R.; Buckmelter, A. J.; Clodfelter, K. H.; Dragovich, P.; Han, B.; Lin, J.; Liu, X.; Reynolds, D. J.; Smith, C. C.; Wang, Z.; Yuen, P-W; Zak, M.; Zhang, Y.; Zhao, G.; Zheng, X. “Amido-benzyl sulfone and sulfonamide derivatives” WO 2013127268, 2013.

  11. Bair, K. W.; Baumeister, T. R.; Dragovich, P.; Gosselin, F.; Yuen, P-W.; Zak, M.; Zheng, X. “Pyridinyl and pyrimidinyl sulfoxide and sulfone derivatives” WO 2013127267, 2013.